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Question

Pharmaceutical Chemistry Question on Different classes of therapeutic drugs

Vigabatrin produces anti-epileptic activity through

A

Potentiating GABA mediated neuronal inhibition by depressing GABA transporters

B

Modifying synaptic release of glutamate/GABA by binding to a specific synaptic protein

C

Inhibiting GABA transaminase enzyme which degrades GABA

D

Potentiating post synaptic GABA receptor effect

Answer

Inhibiting GABA transaminase enzyme which degrades GABA

Explanation

Solution

The correct option is (C): Inhibiting GABA transaminase enzyme which degrades GABA