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Question

Pharmacology Question on Drug therapy

Imipenem,a newer antibiotic with a broad antibacterial spectrum, is co administered with cilastatin. Which of the following is the best reason for the same?

A

Combination of antibiotics is synergistic against Pseudomonas specie

B

Cilastatin aids gastrointestinal absorption of active moiety, imipenem

C

Cilastatin inhibits beta=lactamase enzyme destroying imipenem

D

Cilastatin inhibits an enzyme in kidney destroying imipenem

Answer

Cilastatin inhibits an enzyme in kidney destroying imipenem

Explanation

Solution

The correct option is (D) : Cilastatin inhibits an enzyme in kidney destroying imipenem