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Question

Pharmaceutical Chemistry Question on Different classes of therapeutic drugs

5-Fluorouracil, an anti-metabolite used in cancer treatment, is activated to:

A

5-fluoro-2-oxyuridylic acid

B

3-fluoro-3-deoxyuridylic acid

C

3-fluoro-3-oxyuridylic acid

D

5-fluoro-2-deoxyuridylic acid

Answer

5-fluoro-2-deoxyuridylic acid

Explanation

Solution

The correct option is (D): 5-fluoro-2-deoxyuridylic acid.